Hexarelin
10 mg (lyophilized)
Purity:
≥99% (HPLC)

Cap colour is for illustration purposes only
Hexarelin
10 mg (lyophilized)
+ $25 flat-rate shipping · free at $300+ · Interac e-Transfer ·
About this compound
Hexarelin is a synthetic hexapeptide growth hormone secretagogue (GHS) and potent agonist of the growth hormone secretagogue receptor (GHSR-1a). Structurally derived from Met-enkephalin, it was one of the first synthetic GHS peptides developed and has been extensively studied in preclinical research for its ability to stimulate pulsatile GH release from the anterior pituitary. Beyond GH secretagogue activity, hexarelin has been investigated for direct cardiovascular effects through its binding to the CD36 scavenger receptor and GHSR-independent cardiac mechanisms, making it a notable compound for multi-pathway preclinical research.
Storage and handling
Store at -20°C lyophilized, away from moisture and UV light. Keep vials sealed until use. Stable for 2+ years in a non-frost-free freezer.
Preclinical research references
Provided for informational context only. All cited studies involve preclinical or in vitro models. Results do not predict human safety or efficacy. These references do not constitute medical claims.
- Rat models demonstrated potent, dose-dependent GH release following subcutaneous and intravenous administration, with peak plasma GH levels significantly exceeding those produced by GHRH alone (Ghigo et al., 1994)
- Rodent cardiac studies observed that hexarelin exerted direct cardioprotective effects independent of GH/IGF-1 elevation, attenuating ischemia-reperfusion injury via CD36 receptor binding in isolated heart models (Bisi et al., 1999)
- Animal research showed hexarelin administration reduced cardiomyocyte apoptosis and improved left ventricular function in rat heart failure models, suggesting GHSR-independent myocardial protective pathways (Tivesten et al., 2000)
- Mouse models demonstrated that repeated hexarelin dosing modulated hypothalamic somatostatin tone, influencing GH secretion feedback and pulsatility patterns across extended study periods (Loche et al., 1995)
Shipping & returns
1–5 business days (5–7 for BC, NL and remote areas), Canada-wide tracked courier, double tamper-proof packaging.
All sales final. Damaged or incorrect orders must be reported within 24 hours with photos.
Every batch independently tested for purity. COA on file and available before purchase.
FAQ — Hexarelin
For research use only. Not for human or veterinary administration.
